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(S)-AM1241
Numer katalogowy: 931-T38147-50mg
Kategoria produktu: Biznes i przemysł > Badania naukowe i laboratoryjne
Sprzedawca:Gentaur
Rozmiar:
50mg
Dostępność:
Na zamówienie
Cena:
0.01 PLN*
* Zapytaj o ofertę, aby otrzymać aktualną ofertę w 24h.
(S)-AM1241
Dodatkowe informacje:
- SMILES: C(=O)(C=1C=2C(N(C[C@H]3N(C)CCCC3)C1)=CC=CC2)C4=CC(N(=O)=O)=CC=C4I
- Formula: C22H22IN3O3
Specyfikacja/Zawartość:
- Purity: 0.98
- CAS#: 444912-53-2
- Molecular Weight: 503.33
- Bioactivity: (S)-AM1241 binds to cannabinoid (CB) receptors and is selective for the CB2 over the CB1 receptor (Kis = 658 and >10,000 nM, respectively, in a membrane assay using human receptors). (S)-1241 acts as an agonist at human, rat, and mouse CB2 receptors but shows greater activity at human CB2 (EC50 = 131 nM) than at rat and mouse CB2 receptors (EC50 = 785 and 2,000 nM, respectively). Similar to the racemate AM1241 , (S)-AM1241 produces antinociception to thermal, but not mechanical, pain in rats. The pain-reducing effect of (S)-AM1241 is blocked by the CB2-specific inhibitor SR 144528 but not by either the CB1-selective inhibitor rimonabant or the opioid receptor blocker naloxone .
Inne:
For research use only.
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